Drug Classes and Mechanisms · USMLE Step 1

Which class of antihypertensives works by blocking angiotensin II from binding to its AT₁ receptor, without affecting bradykinin metabolism?

  1. ACE inhibitors
  2. Beta-blockers
  3. ARBs
  4. Thiazide diuretics
Show answer and explanation

Correct answer: ARBs

Angiotensin II receptor blockers (ARBs) competitively inhibit binding of angiotensin II to AT₁ receptors, leading to vasodilation and BP reduction without altering bradykinin levels.

Difficulty: Medium Question 4 of 19

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