Drug Classes and Mechanisms · USMLE Step 1

Which drug class lowers heart rate and myocardial contractility primarily by antagonizing β₁-adrenergic receptors in the heart?

  1. ACE inhibitors
  2. Calcium channel blockers
  3. Beta-blockers
  4. Diuretics
Show answer and explanation

Correct answer: Beta-blockers

Beta-blockers antagonize β₁-adrenergic receptors in the heart, reducing heart rate and contractility, thereby decreasing cardiac output and blood pressure.

Difficulty: Medium Question 6 of 19

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