Sedatives and Hypnotics · Pharmacology

Suvorexant represents a newer class of hypnotics that works by which mechanism?

  1. Activation of melatonin (MT1 and MT2) receptors
  2. Antagonism of orexin (hypocretin) receptors
  3. Partial agonism of 5-HT1A receptors
  4. Irreversible inhibition of GABA transaminase
Show answer and explanation

Correct answer: Antagonism of orexin (hypocretin) receptors

Suvorexant is a Dual Orexin Receptor Antagonist (DORA). It promotes sleep by blocking the 'wake-promoting' neuropeptides orexin A and B from binding to their receptors, effectively turning off the brain's arousal system.

Difficulty: Medium Question 6 of 20

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