Cholinergic Agonists · Pharmacology

Pilocarpine is frequently used in ophthalmology to treat glaucoma. What is its primary effect on the eye?

  1. Mydriasis and increased intraocular pressure
  2. Mydriasis and decreased intraocular pressure
  3. Miosis and increased intraocular pressure
  4. Miosis and decreased intraocular pressure
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Correct answer: Miosis and decreased intraocular pressure

Pilocarpine stimulates muscarinic receptors on the pupillary constrictor muscle, causing miosis, and on the ciliary muscle, causing contraction. This opens the trabecular meshwork, facilitating the drainage of aqueous humor and lowering intraocular pressure.

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