Chemotherapy and Toxicology · USMLE Step 1

Which antimetabolite is most likely to cause hepatotoxicity and requires careful monitoring of liver enzymes?

  1. Methotrexate
  2. Vinblastine
  3. Cisplatin
  4. Bleomycin
Show answer and explanation

Correct answer: Methotrexate

Methotrexate is metabolized by the liver and can cause hepatotoxicity; many antimetabolites are processed by hepatic pathways making the liver vulnerable.

Difficulty: Medium Question 15 of 20

Practice all 20 Chemotherapy and Toxicology questions

Keep practicing

More Chemotherapy and Toxicology questions