Local Anesthetics · Pharmacology

Which factor mainly determines the duration of action of a local anesthetic?

  1. Lipid solubility
  2. Molecular size
  3. Protein binding
  4. pKa of the drug
Show answer and explanation

Correct answer: Protein binding

Drugs with higher protein binding tend to remain attached to sodium channels longer. This prolongs their duration of anesthetic action.

Difficulty: Medium Question 15 of 20

Practice all 20 Local Anesthetics questions

Keep practicing

More Local Anesthetics questions