Megaloblastic Anemia · Pathology

Which of the following drugs is a known dihydrofolate reductase inhibitor that can cause megaloblastic changes?

  1. Penicillin
  2. Methotrexate
  3. Warfarin
  4. Aspirin (acetylsalicylic acid)
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Correct answer: Methotrexate

Methotrexate is a folate antagonist that inhibits dihydrofolate reductase, the enzyme responsible for regenerating active folate. This interference with the folate cycle inhibits DNA synthesis and can lead to megaloblastic anemia.

Difficulty: Medium Question 10 of 20

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