Drug Classes and Mechanisms · USMLE Step 1

Which drug class lowers blood pressure via direct relaxation of vascular smooth muscle rather than altering renal sodium excretion or hormonal pathways?

  1. ACE inhibitors
  2. Beta-blockers
  3. Calcium channel blockers
  4. Loop diuretics
Show answer and explanation

Correct answer: Calcium channel blockers

Calcium channel blockers act directly on vascular smooth muscle by blocking calcium influx, causing vasodilation independent of renal or hormonal mechanisms.

Difficulty: Medium Question 14 of 19

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