Bronchodilators · Pharmacology

Which enzyme's metabolism is a major concern for Theophylline, leading to numerous drug-drug interactions?

  1. CYP2D6
  2. CYP1A2
  3. Monoamine oxidase
  4. Alcohol dehydrogenase
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Correct answer: CYP1A2

Theophylline is primarily metabolized by CYP1A2. Drugs that inhibit this enzyme (like ciprofloxacin) or induce it (like cigarette smoke) can cause toxic or sub-therapeutic levels, respectively.

Difficulty: Medium Question 7 of 20

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