Half-Life and Clearance · Pharmacology

If a drug has a very short half-life (e.g., 2 minutes) and requires a sustained effect, what is the most appropriate route of administration?

  1. Oral tablet once daily
  2. Subcutaneous injection every 12 hours
  3. Continuous intravenous infusion
  4. Single intramuscular bolus
Show answer and explanation

Correct answer: Continuous intravenous infusion

Drugs with very short half-lives, like esmolol or nitroglycerin, are eliminated too quickly for intermittent dosing. A continuous infusion allows for minute-to-minute control of plasma levels and sustained therapeutic action.

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