Stimulants · Pharmacology

Which stimulant mechanism directly increases synaptic dopamine concentration?

  1. Inhibition of dopamine reuptake
  2. Activation of GABA receptors
  3. Blocking sodium channels
  4. Inhibition of acetylcholine release
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Correct answer: Inhibition of dopamine reuptake

Stimulants such as methylphenidate increase synaptic dopamine by inhibiting its reuptake. This prolongs dopaminergic signaling and enhances alertness.

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