Stimulants · Pharmacology

Caffeine exerts its stimulant effect primarily by:

  1. Enhancing GABA activity
  2. Blocking adenosine receptors
  3. Inhibiting monoamine oxidase
  4. Stimulating opioid receptors
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Correct answer: Blocking adenosine receptors

Caffeine acts as an antagonist at adenosine receptors. By blocking adenosine’s inhibitory effects, it increases neuronal firing and alertness.

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