Liver and Pancreas Functions · Physiology

Phase I of hepatic drug metabolism typically involves which of the following chemical modifications?

  1. Conjugation of the drug with glutathione
  2. Oxidation or reduction via cytochrome P450
  3. Attachment of a glucuronide group to the drug
  4. Sulfation of the drug molecule for excretion
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Correct answer: Oxidation or reduction via cytochrome P450

Phase I reactions (functionalization) usually involve the Cytochrome P450 system to add or expose a polar group. Phase II reactions involve conjugation, where a large polar molecule is attached to make the drug ready for excretion.

Difficulty: Medium Question 39 of 40

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